β-榄香烯是从天然药用植物温莪术中提取的萜烯类有效活性成分，具有分子质量小、抗肿瘤强、毒性低等特点，临床上用于非小细胞肺癌（on-small-cell lung cancer，NSCLC）常规治疗的辅助用药。β-榄香烯能通过抑制肿瘤细胞增殖，诱导肿瘤细胞凋亡，抑制肿瘤血管形成，阻滞细胞周期，逆转耐药，以及调节免疫能力等发挥抗肿瘤作用。基于榄香烯已有研究基础，对其抑制NSCLC作用机制的研究进展进行综述，以期为临床上更好地将榄香烯用于NSCLC辅助支持治疗提供理论依据和思路。

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